Bisnortilidine

Bisnortilidine
Names
IUPAC name
Ethyl (1R,2S)-2-amino-1-phenylcyclohex-3-ene-1-carboxylate
Identifiers
ChemSpider 454879
Jmol interactive 3D Image
PubChem 162740
Properties
C15H19NO2
Molar mass 245.32 g·mol−1
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
Infobox references

Bisnortilidine is an opioid metabolite.[1] It is formed from tilidine by demethylation in the liver.

References

  1. Wustrow, I.; Riedel, K. D.; Mikus, G.; Weiss, J. (2012). "In vitro identification of the cytochrome P450 isozymes involved in the N-demethylation of the active opioid metabolite nortilidine to bisnortilidine". Naunyn-Schmiedeberg's Archives of Pharmacology 385 (6): 633–9. doi:10.1007/s00210-012-0737-z. PMID 22349139.


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