Cicloprolol

Cicloprolol

Names
IUPAC name 1-[4-[2-(Cyclopropylmethoxy)ethoxy]phenoxy]-3-(propan-2-ylamino)propan-2-ol
Identifiers
CAS Number	91094-14-3
ChEMBL	ChEMBL2110772
ChemSpider	129044
IUPHAR/BPS	552
Jmol interactive 3D	Image
PubChem	146294
InChI InChI=1S/C18H29NO4/c1-14(2)19-11-16(20)13-23-18-7-5-17(6-8-18)22-10-9-21-12-15-3-4-15/h5-8,14-16,19-20H,3-4,9-13H2,1-2H3 Key: JNDJPKHYZWRRIS-UHFFFAOYSA-N
SMILES CC(C)NCC(COC1=CC=C(C=C1)OCCOCC2CC2)O
Properties
Chemical formula	C18H29NO4
Molar mass	323.43 g·mol^−1
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
Infobox references

Cicloprolol is a beta-adrenoceptor antagonist.^[1]

Synthesis

Cicloprolol synthesis:^[2]

See also

• Betaxolol

References

1. Cocco, G; Alfiero, R; Pouleur, H (1992). "An evaluation of the safety of the beta-modulator cicloprolol in chronic heart failure". Clinical Cardiology 15 (1): 38–42. doi:10.1002/clc.4960150109. PMID 1347258.
2. P. M. J. Manouri, I. A. G. Carero, H. Majer, and P. R. L. Giudicelli, DE 2649605  (1977) via Chem. Abstr., 87:134,543j (1977). eidem U.S. Patent 4,311,708