Latrunculin
Chemical structures of latrunculins
The latrunculins are a family of natural products and toxins produced by certain sponges, including genus Latrunculia and Negombata, whence the name is derived. It binds actin monomers near the nucleotide binding cleft with 1:1 stoichiometry and prevents them from polymerizing. Administered in vivo, this effect results in disruption of the actin filaments of the cytoskeleton. This property has been used to great effect in the discovery of cadherin distribution regulation.
References
- Yarmola, E.G., Somasundaram, T., Boring, T.A., Spector, I., Bubb, M.R. (2000). "Actin-Latrunculin A Structure and Function". Journal of Biological Chemistry 275 (36): 28120–28127. doi:10.1074/jbc.M004253200. PMID 10859320.
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