Timepidium bromide

Timepidium bromide
Systematic (IUPAC) name

3-(di-2-thienylmethylene)-5-methoxy-1,1-dimethylpiperidinium bromide
Clinical data
AHFS/Drugs.com	International Drug Names
Routes of administration	SC, IM, IV
Legal status
Legal status	℞ (Prescription only)
Identifiers
CAS Number	35035-05-3^Y
ATC code	A03AB19 (WHO)
PubChem	CID 160243
ChemSpider	140841^N
UNII	8R9E4766V4^N
Chemical data
Formula	C₁₇H₂₂BrNOS₂
Molar mass	400.39 g/mol
SMILES C[N+]1(CC(CC(=C(C2=CC=CS2)C3=CC=CS3)C1)OC)C.[Br-]
InChI InChI=1S/C17H22NOS2.BrH/c1-18(2)11-13(10-14(12-18)19-3)17(15-6-4-8-20-15)16-7-5-9-21-16;/h4-9,14H,10-12H2,1-3H3;1H/q+1;/p-1^N Key:QTSXMEPZSHLZFF-UHFFFAOYSA-M^N
^NY (what is this?) (verify)

Timepidium bromide (INN) is an anticholinergic. The quaternary nitrogen prevents it from crossing the blood brain barrier, so it is peripherally acting with no central side effects.

The same compound sans the quaternary methyl group and the methoxy ether is called tipepidine.

Drugs for functional gastrointestinal disorders (A03)

Drugs for
functional
bowel disorders

Antimuscarinics

Tertiary amino group	Oxyphencyclimine Camylofin Mebeverine Trimebutine Rociverine Dicycloverine Dihexyverine Difemerine Piperidolate

Quaternary ammonium compounds	Benzilone Mepenzolate Pipenzolate Glycopyrronium Oxyphenonium Penthienate Methantheline Propantheline Otilonium Tridihexethyl Isopropamide Hexocyclium Poldine Bevonium Diphemanil Tiemonium Prifinium Timepidium Fenpiverinium

Phosphodiesterase
inhibitors

Acting on
serotonin receptors

Other

Belladonna
and derivatives
(antimuscarinics)

tertiary amines: Atropine
Hyoscyamine

Propulsives

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