| Name | Trade name | Type | Source | Target | Use |
| 3F8 | | mab | mouse | GD2 | neuroblastoma |
| 8H9[1] | | mab | mouse | B7-H3 | neuroblastoma, sarcoma, metastatic brain cancers |
| Abagovomab[2] | | mab | mouse | CA-125 (imitation) | ovarian cancer |
| Abciximab | ReoPro | Fab | chimeric | CD41 (integrin alpha-IIb) | platelet aggregation inhibitor |
| Abituzumab[3] | | mab | humanized | CD51 | cancer |
| Abrilumab[4] | | mab | human | integrin α4β7 | inflammatory bowel disease, ulcerative colitis, Crohn's disease |
| Actoxumab[5] | | mab | human | Clostridium difficile | Clostridium difficile colitis |
| Adalimumab | Humira | mab | human | TNF-α | Rheumatoid arthritis, Crohn's Disease, Plaque Psoriasis, Psoriatic Arthritis, Ankylosing Spondylitis, Juvenile Idiopathic Arthritis, Hemolytic disease of the newborn |
| Adecatumumab[6] | | mab | human | EpCAM | prostate and breast cancer |
| Aducanumab[7] | | mab | human | beta-amyloid | Alzheimer's disease |
| Afelimomab | | F(ab')2 | mouse | TNF-α | sepsis |
| Afutuzumab[8] | | mab | humanized | CD20 | lymphoma |
| Alacizumab pegol[9] | | F(ab')2 | humanized | VEGFR2 | cancer |
| ALD518[10] | | ? | humanized | IL-6 | rheumatoid arthritis |
| Alemtuzumab[11] | Lemtrada, Campath | mab | humanized | CD52 | Multiple sclerosis |
| Alirocumab[12] | | mab | human | PCSK9 | hypercholesterolemia |
| Altumomab pentetate | Hybri-ceaker | mab | mouse | CEA | colorectal cancer (diagnosis) |
| Amatuximab[13] | | mab | chimeric | mesothelin | cancer |
| Anatumomab mafenatox | | Fab | mouse | TAG-72 | non-small cell lung carcinoma |
| Anetumab ravtansine[3] | | mab | human | MSLN | cancer |
| Anifrolumab[14] | | mab | human | interferon α/β receptor | systemic lupus erythematosus |
| Anrukinzumab[9] (= IMA-638)[15] | | mab | humanized | IL-13 | ? |
| Apolizumab[16] | | mab | humanized | HLA-DR ? | hematological cancers |
| Arcitumomab | CEA-Scan | Fab' | mouse | CEA | gastrointestinal cancers (diagnosis) |
| Ascrinvacumab[17] | | mab | human | activin receptor-like kinase 1 | cancer |
| Aselizumab[18] | | mab | humanized | L-selectin (CD62L) | severely injured patients |
| Atezolizumab[19] | | mab | humanized | CD274 | cancer |
| Atinumab[20] | | mab | human | RTN4 | ? |
| Atlizumab (= tocilizumab) | Actemra, RoActemra | mab | humanized | IL-6 receptor | rheumatoid arthritis |
| Atorolimumab | | mab | human | Rhesus factor | hemolytic disease of the newborn |
| Bapineuzumab[21] | | mab | humanized | beta amyloid | Alzheimer's disease |
| Basiliximab | Simulect | mab | chimeric | CD25 (α chain of IL-2 receptor) | prevention of organ transplant rejections |
| Bavituximab[2] | | mab | chimeric | phosphatidylserine | cancer, viral infections |
| Bectumomab | LymphoScan | Fab' | mouse | CD22 | non-Hodgkin's lymphoma (detection) |
| Begelomab[22] | | mab | mouse | DPP4 | ? |
| Belimumab | Benlysta, LymphoStat-B | mab | human | BAFF | non-Hodgkin lymphoma etc. |
| Benralizumab | | mab | humanized | CD125 | asthma |
| Bertilimumab[18] | | mab | human | CCL11 (eotaxin-1) | severe allergic disorders |
| Besilesomab[23] | Scintimun | mab | mouse | CEA-related antigen | inflammatory lesions and metastases (detection) |
| Bevacizumab[11] | Avastin | mab | humanized | VEGF-A | metastatic cancer, retinopathy of prematurity |
| Bezlotoxumab[24] | | mab | human | Clostridium difficile | Clostridium difficile colitis |
| Biciromab | FibriScint | Fab' | mouse | fibrin II, beta chain | thromboembolism (diagnosis) |
| Bimagrumab[25][26] | | mab | human | ACVR2B | myostatin inhibitor |
| Bimekizumab[27] | | mab | humanized | IL 17A and IL 17F | ? |
| Bivatuzumab mertansine | | mab | humanized | CD44 v6 | squamous cell carcinoma |
| Blinatumomab | | BiTE | mouse | CD19 | cancer |
| Blosozumab[28] | | mab | humanized | SOST | osteoporosis |
| Bococizumab[29] | | mab | humanized | neural apoptosis-regulated proteinase 1 | dyslipidemia |
| Brentuximab vedotin[30] | | mab | chimeric | CD30 (TNFRSF8) | hematologic cancers |
| Briakinumab[31] | | mab | human | IL-12, IL-23 | psoriasis, rheumatoid arthritis, inflammatory bowel diseases, multiple sclerosis |
| Brodalumab[32] | | mab | human | IL-17 | inflammatory diseases |
| Brolucizumab[19] | | mab | humanized | VEGFA | ? |
| Brontictuzumab[22] | | mab | Notch 1 | cancer |
| Canakinumab[33] | Ilaris | mab | human | IL-1? | rheumatoid arthritis |
| Cantuzumab mertansine | | mab | humanized | mucin CanAg | colorectal cancer etc. |
| Cantuzumab ravtansine[28] | | mab | humanized | MUC1 | cancers |
| Caplacizumab[34] | | mab | humanized | VWF | thrombotic thrombocytopenic purpura, thrombosis |
| Capromab pendetide | Prostascint | mab | mouse | prostatic carcinoma cells | prostate cancer (detection) |
| Carlumab[35] | | mab | human | MCP-1 | oncology/immune indications |
| Catumaxomab[21] | Removab | 3funct | rat/mouse hybrid | EpCAM, CD3 | ovarian cancer, malignant ascites, gastric cancer |
| cBR96-doxorubicin immunoconjugate | | mab | humanized | Lewis-Y antigen | cancer |
| Cedelizumab | | mab | humanized | CD4 | prevention of organ transplant rejections, treatment of autoimmune diseases |
| Certolizumab pegol[6] | Cimzia | Fab' | humanized | TNF-α | Crohn's disease |
| Cetuximab | Erbitux | mab | chimeric | EGFR | metastatic colorectal cancer and head and neck cancer |
| Ch.14.18 [1] | | mab | chimeric | ??? | neuroblastoma |
| Citatuzumab bogatox[8] | | Fab | humanized | EpCAM | ovarian cancer and other solid tumors |
| Cixutumumab | | mab | human | IGF-1 receptor | solid tumors |
| Clazakizumab[36] | | mab | humanized | Oryctolagus cuniculus | rheumatoid arthritis |
| Clenoliximab | | mab | chimeric | CD4 | rheumatoid arthritis |
| Clivatuzumab tetraxetan[37] | hPAM4-Cide | mab | humanized | MUC1 | pancreatic cancer |
| Codrituzumab[3] | | mab | humanized | glypican 3 | cancer |
| Coltuximab ravtansine[3] | | mab | chimeric | CD19 | cancer |
| Conatumumab[8] | | mab | human | TRAIL-R2 | cancer |
| Concizumab[25] | | mab | humanized | TFPI | bleeding |
| Crenezumab[38] | | mab | humanized | 1-40-β-amyloid | Alzheimer's disease |
| CR6261 | | mab | human | Influenza A hemagglutinin | infectious disease/influenza A |
| Dacetuzumab[9] | | mab | humanized | CD40 | hematologic cancers |
| Daclizumab | Zenapax | mab | humanized | CD25 (α chain of IL-2 receptor) | prevention of organ transplant rejections |
| Dalotuzumab[39] | | mab | humanized | insulin-like growth factor I receptor | cancer etc. |
| Dapirolizumab pegol[27] | | mab | humanized | CD40 ligand | ? |
| Daratumumab[40] | | mab | human | CD38 (cyclic ADP ribose hydrolase) | cancer |
| Dectrekumab[19] | | mab | human | IL-13 | ? |
| Demcizumab[41] | | mab | humanized | DLL4 | cancer |
| Denintuzumab mafodotin[22] | | mab | humanized | CD19 | cancer |
| Denosumab[42] | Prolia | mab | human | RANKL | osteoporosis, bone metastases etc. |
| Derlotuximab biotin[43] | | mab | chimeric | histone complex | recurrent glioblastoma multiforme |
| Detumomab | | mab | mouse | B-lymphoma cell | lymphoma |
| Dinutuximab[44] | | mab | chimeric | ganglioside GD2 | neuroblastoma |
| Diridavumab[45] | | mab | human | hemagglutinin | influenza A |
| Dorlimomab aritox[46] | | F(ab')2 | mouse | ? | ? |
| Drozitumab[47] | | mab | human | DR5 | cancer etc. |
| Duligotumab[48] | | mab | human | HER3 | ? |
| Dupilumab[49] | | mab | human | IL4 | atopic diseases |
| Durvalumab[50] | | mab | human | CD274 | cancer |
| Dusigitumab[51] | | mab | human | ILGF2 | cancer |
| Ecromeximab[16] | | mab | chimeric | GD3 ganglioside | malignant melanoma |
| Eculizumab[16] | Soliris | mab | humanized | C5 | paroxysmal nocturnal hemoglobinuria |
| Edobacomab | | mab | mouse | endotoxin | sepsis caused by Gram-negative bacteria |
| Edrecolomab | Panorex | mab | mouse | EpCAM | colorectal carcinoma |
| Efalizumab[52] | Raptiva | mab | humanized | LFA-1 (CD11a) | psoriasis (blocks T-cell migration) |
| Efungumab[2] | Mycograb | scFv | human | Hsp90 | invasive Candida infection |
| Eldelumab[53] | | mab | human | interferon gamma-induced protein | Crohn's disease, ulcerative colitis |
| Elgemtumab[19] | | mab | human | ERBB3 | cancer |
| Elotuzumab | | mab | humanized | SLAMF7 | multiple myeloma |
| Elsilimomab | | mab | mouse | IL-6 | ? |
| Emactuzumab[22] | | mab | humanized | CSF1R | cancer |
| Emibetuzumab[54] | | mab | humanized | HHGFR | cancer |
| Enavatuzumab[55] | | mab | humanized | TWEAK receptor | cancer etc. |
| Enfortumab vedotin[56] | | mab | human | AGS-22M6 | cancer expressing Nectin-4 |
| Enlimomab pegol[57] | | mab | mouse | ICAM-1 (CD54) | ? |
| Enoblituzumab[58] | | mab | humanized | B7-H3 | cancer |
| Enokizumab[59] | | mab | humanized | IL9 | asthma |
| Enoticumab[48] | | mab | human | DLL4 | ? |
| Ensituximab[60] | | mab | chimeric | 5AC | cancer |
| Epitumomab cituxetan[61] | | mab | mouse | episialin | ? |
| Epratuzumab | | mab | humanized | CD22 | cancer, SLE |
| Erlizumab[62] | | F(ab')2 | humanized | ITGB2 (CD18) | heart attack, stroke, traumatic shock |
| Ertumaxomab[21] | Rexomun | 3funct | rat/mouse hybrid | HER2/neu, CD3 | breast cancer etc. |
| Etaracizumab | Abegrin | mab | humanized | integrin αvβ3 | melanoma, prostate cancer, ovarian cancer etc. |
| Etrolizumab[63] | | mab | humanized | integrin α7 β7 | inflammatory bowel disease |
| Evinacumab[64] | | mab | human | angiopoietin 3 | dyslipidemia |
| Evolocumab[25] | | mab | human | PCSK9 | hypercholesterolemia |
| Exbivirumab[65] | | mab | human | hepatitis B surface antigen | hepatitis B |
| Fanolesomab[66] | NeutroSpec | mab | mouse | CD15 | appendicitis (diagnosis) |
| Faralimomab | | mab | mouse | interferon receptor | ? |
| Farletuzumab | | mab | humanized | folate receptor 1 | ovarian cancer |
| Fasinumab[67] | | mab | human | HNGF | acute sciatic pain |
| FBTA05[68][69] | Lymphomun | 3funct | rat/mouse hybrid | CD20 | chronic lymphocytic leukaemia |
| Felvizumab | | mab | humanized | respiratory syncytial virus | respiratory syncytial virus infection |
| Fezakinumab[70][71][72] | | mab | human | IL-22 | rheumatoid arthritis, psoriasis |
| Ficlatuzumab[73] | | mab | humanized | HGF | cancer etc. |
| Figitumumab | | mab | human | IGF-1 receptor | adrenocortical carcinoma, non-small cell lung carcinoma etc. |
| Firivumab[22] | | mab | human | influenza A virus hemagglutinin | ? |
| Flanvotumab[74] | | mab | human | TYRP1(glycoprotein 75) | melanoma |
| Fletikumab[75] | | mab | human | IL 20 | rheumatoid arthritis |
| Fontolizumab[16] | HuZAF | mab | humanized | IFN-γ | Crohn's disease etc. |
| Foralumab[76] | | mab | human | CD3 epsilon | ? |
| Foravirumab[8] | | mab | human | rabies virus glycoprotein | rabies (prophylaxis) |
| Fresolimumab[77] | | mab | human | TGF-β | idiopathic pulmonary fibrosis, focal segmental glomerulosclerosis, cancer |
| Fulranumab[78] | | mab | human | NGF | pain |
| Futuximab[48] | | mab | chimeric | EGFR | ? |
| Galiximab | | mab | chimeric | CD80 | B-cell lymphoma |
| Ganitumab[79] | | mab | human | IGF-I | cancer |
| Gantenerumab[33] | | mab | human | beta amyloid | Alzheimer's disease |
| Gavilimomab[62] | | mab | mouse | CD147 (basigin) | graft versus host disease |
| Gemtuzumab ozogamicin | Mylotarg | mab | humanized | CD33 | acute myelogenous leukemia |
| Gevokizumab[80] | | mab | humanized | IL-1β | diabetes etc. |
| Girentuximab[40] | Rencarex | mab | chimeric | carbonic anhydrase 9 (CA-IX) | clear cell renal cell carcinoma[81] |
| Glembatumumab vedotin[82][83] | | mab | human | GPNMB | melanoma, breast cancer |
| Golimumab[65] | Simponi | mab | human | TNF-α | rheumatoid arthritis, psoriatic arthritis, ankylosing spondylitis |
| Gomiliximab | | mab | chimeric | CD23 (IgE receptor) | allergic asthma |
| Guselkumab[84] | | mab | human | IL23 | psoriasis |
| Ibalizumab[33] | | mab | humanized | CD4 | HIV infection |
| Ibritumomab tiuxetan | Zevalin | mab | mouse | CD20 | non-Hodgkin's lymphoma |
| Icrucumab[85] | | mab | human | VEGFR-1 | cancer etc. |
| Idarucizumab[3] | | mab | humanized | dabigatran | reversal of anticoagulant effects of dabigatran |
| Igovomab | Indimacis-125 | F(ab')2 | mouse | CA-125 | ovarian cancer (diagnosis) |
| IMAB362 | | mab | human | CLDN18.2 | gastrointestinal adenocarcinomas and pancreatic tumor |
| Imalumab[22] | | mab | human | MIF | cancer |
| Imciromab | Myoscint | mab | mouse | cardiac myosin | cardiac imaging |
| Imgatuzumab[48] | | mab | humanized | EGFR | cancer |
| Inclacumab[34] | | mab | human | selectin P | ? |
| Indatuximab ravtansine[28] | | mab | chimeric | SDC1 | cancer |
| Indusatumab vedotin[19] | | mab | human | GUCY2C | cancer |
| Infliximab | Remicade | mab | chimeric | TNF-α | rheumatoid arthritis, ankylosing spondylitis, psoriatic arthritis, psoriasis, Crohn's disease, ulcerative colitis |
| Intetumumab[86][87][88] | | mab | human | CD51 | solid tumors (prostate cancer, melanoma) |
| Inolimomab | | mab | mouse | CD25 (α chain of IL-2 receptor) | graft versus host disease |
| Inotuzumab ozogamicin[23] | | mab | humanized | CD22 | cancer |
| Ipilimumab[42] | Yervoy | mab | human | CD152 | melanoma |
| Iratumumab[42] | | mab | human | CD30 (TNFRSF8) | Hodgkin's lymphoma |
| Isatuximab[89] | | mab | chimeric | CD38 | cancer |
| Itolizumab[76] | | mab | humanized | CD6 | ? |
| Ixekizumab[90] | | mab | humanized | IL 17A | autoimmune diseases |
| Keliximab | | mab | chimeric | CD4 | chronic asthma |
| Labetuzumab[52] | CEA-Cide | mab | humanized | CEA | colorectal cancer |
| Lambrolizumab[91] | | mab | humanized | PDCD1 | antineoplastic agent |
| Lampalizumab[48] | | mab | humanized | CFD | ? |
| Lebrikizumab[92] | | mab | humanized | IL-13 | asthma |
| Lemalesomab[62] | | mab | mouse | NCA-90 (granulocyte antigen) | diagnostic agent |
| Lenzilumab[22] | | mab | human | CSF2 | ? |
| Lerdelimumab[11] | | mab | human | TGF beta 2 | reduction of scarring after glaucoma surgery |
| Lexatumumab[2] | | mab | human | TRAIL-R2 | cancer |
| Libivirumab[65] | | mab | human | hepatitis B surface antigen | hepatitis B |
| Lifastuzumab vedotin[93] | | mab | humanized | phosphate-sodium co-transporter | cancer |
| Ligelizumab[48][94] | | mab | humanized | IGHE | severe asthma and chronic spontaneous urticaria |
| Lilotomab satetraxetan[19] | | mab | mouse | CD37 | cancer |
| Lintuzumab | | mab | humanized | CD33 | cancer |
| Lirilumab[48] | | mab | human | KIR2D | ? |
| Lodelcizumab[25] | | mab | humanized | PCSK9 | hypercholesterolemia |
| Lokivetmab[19] | | mab | veterinary | Canis lupus familiaris IL31 | ? |
| Lorvotuzumab mertansine | | mab | humanized | CD56 | cancer |
| Lucatumumab[9] | | mab | human | CD40 | multiple myeloma, non-Hodgkin's lymphoma, Hodgkin's lymphoma |
| Lulizumab pegol[95] | | mab | humanized | CD28 | autoimmune diseases |
| Lumiliximab[6] | | mab | chimeric | CD23 (IgE receptor) | chronic lymphocytic leukemia |
| Lumretuzumab[22] | | mab | humanized | ERBB3 | cancer |
| Mapatumumab[21] | | mab | human | TRAIL-R1 | cancer |
| Margetuximab[96] | | mab | humanized | ch4D5 | cancer |
| Maslimomab | | ? | mouse | T-cell receptor | ? |
| Mavrilimumab[97] | | mab | human | GMCSF receptor α-chain | rheumatoid arthritis |
| Matuzumab[18] | | mab | humanized | EGFR | colorectal, lung and stomach cancer |
| Mepolizumab | Bosatria | mab | humanized | IL-5 | asthma and white blood cell diseases |
| Metelimumab[66] | | mab | human | TGF beta 1 | systemic scleroderma |
| Milatuzumab[9] | | mab | humanized | CD74 | multiple myeloma and other hematological malignancies |
| Minretumomab | | mab | mouse | TAG-72 | tumor detection (and therapy?) |
| Mirvetuximab soravtansine[98] | | mab | chimeric | folate receptor alpha | cancer |
| Mitumomab | | mab | mouse | GD3 ganglioside | small cell lung carcinoma |
| Mogamulizumab[99] | | mab | humanized | CCR4 | cancer |
| Morolimumab | | mab | human | Rhesus factor | ? |
| Motavizumab[2] | Numax | mab | humanized | respiratory syncytial virus | respiratory syncytial virus (prevention) |
| Moxetumomab pasudotox[100] | | mab | mouse | CD22 | cancer |
| Muromonab-CD3 | Orthoclone OKT3 | mab | mouse | CD3 | prevention of organ transplant rejections |
| Nacolomab tafenatox | | Fab | mouse | C242 antigen | colorectal cancer |
| Namilumab[20] | | mab | human | CSF2 | ? |
| Naptumomab estafenatox[101] | | Fab | mouse | 5T4 | non-small cell lung carcinoma, renal cell carcinoma |
| Narnatumab[102] | | mab | human | RON | cancer |
| Natalizumab | Tysabri | mab | humanized | integrin α4 | multiple sclerosis, Crohn's disease |
| Nebacumab | | mab | human | endotoxin | sepsis |
| Necitumumab[103] | | mab | human | EGFR | non-small cell lung carcinoma |
| Nemolizumab[19] | | mab | humanized | IL31RA | ? |
| Nerelimomab | | mab | mouse | TNF-α | ? |
| Nesvacumab[104] | | mab | human | angiopoietin 2 | cancer |
| Nimotuzumab[42][105] | Theracim, Theraloc | mab | humanized | EGFR | squamous cell carcinoma, head and neck cancer, nasopharyngeal cancer, glioma |
| Nivolumab[106] | Opdivo | mab | human | PD-1 | cancer |
| Nofetumomab merpentan | Verluma | Fab | mouse | ? | cancer (diagnosis) |
| Obiltoxaximab[107] | | mab | chimeric | Bacillus anthracis anthrax | Bacillus anthracis spores |
| Obinutuzumab |
Gazyva |
mab |
humanized |
CD20 |
Chronic lymphatic leukemia |
| Ocaratuzumab[108] | | mab | humanized | CD20 | cancer |
| Ocrelizumab[42] | | mab | humanized | CD20 | rheumatoid arthritis, lupus erythematosus etc. |
| Odulimomab | | mab | mouse | LFA-1 (CD11a) | prevention of organ transplant rejections, immunological diseases |
| Ofatumumab[21] | Arzerra | mab | human | CD20 | chronic lymphocytic leukemia etc. |
| Olaratumab | | mab | human | PDGF-R α | cancer |
| Olokizumab[76] | | mab | humanized | IL6 | ? |
| Omalizumab[62] | Xolair | mab | humanized | IgE Fc region | allergic asthma |
| Onartuzumab[109] | | mab | humanized | human scatter factor receptor kinase | cancer |
| Ontuxizumab[110] | | mab | chimeric/humanized | TEM1 | cancer |
| Opicinumab[111] | | mab | human | LINGO-1 | multiple sclerosis |
| Oportuzumab monatox[103] | | scFv | humanized | EpCAM | cancer |
| Oregovomab[66] | OvaRex | mab | mouse | CA-125 | ovarian cancer |
| Orticumab[48] | | mab | human | oxLDL | ? |
| Otelixizumab[9] | | mab | chimeric/humanized | CD3 | diabetes mellitus type 1 |
| Otlertuzumab[112] | | mab | humanized | CD37 | cancer |
| Oxelumab[113] | | mab | human | OX-40 | asthma |
| Ozanezumab[114] | | mab | humanized | NOGO-A | ALS and multiple sclerosis |
| Ozoralizumab[115] | | mab | humanized | TNF-α | inflammation |
| Pagibaximab[21] | | mab | chimeric | lipoteichoic acid | sepsis (Staphylococcus) |
| Palivizumab | Synagis, Abbosynagis | mab | humanized | F protein of respiratory syncytial virus | respiratory syncytial virus (prevention) |
| Panitumumab[65] | Vectibix | mab | human | EGFR | colorectal cancer |
| Pankomab | | mab | humanized | tumor specific glycosylation of MUC1 | ovarian cancer |
| Panobacumab[103] | | mab | human | Pseudomonas aeruginosa | Pseudomonas aeruginosa infection |
| Parsatuzumab[48] | | mab | human | EGFL7 | cancer |
| Pascolizumab[16] | | mab | humanized | IL-4 | asthma |
| Pasotuxizumab[22] | | mab | chimeric/humanized | folate hydrolase | cancer |
| Pateclizumab[28] | | mab | humanized | LTA | TNF |
| Patritumab[34] | | mab | human | HER3 | cancer |
| Pembrolizumab[116] | | mab | humanized | PDCD1 | cancer etc. |
| Pemtumomab | Theragyn | ? | mouse | MUC1 | cancer |
| Perakizumab[48] | | mab | humanized | IL 17A | arthritis |
| Pertuzumab | Omnitarg | mab | humanized | HER2/neu | cancer |
| Pexelizumab[52] | | scFv | humanized | C5 | reduction of side effects of cardiac surgery |
| Pidilizumab[117] | | mab | humanized | PD-1 | cancer and infectious diseases |
| Pinatuzumab vedotin[25] | | mab | humanized | CD22 | cancer |
| Pintumomab | | mab | mouse | adenocarcinoma antigen | adenocarcinoma (imaging) |
| Placulumab[118] | | mab | human | human TNF | ? |
| Polatuzumab vedotin[25][119] | | mab | humanized | CD79B | cancer |
| Ponezumab[120] | | mab | humanized | human beta-amyloid | Alzheimer's disease |
| Priliximab | | mab | chimeric | CD4 | Crohn's disease, multiple sclerosis |
| Pritoxaximab[25] | | mab | chimeric | E. coli shiga toxin type-1 | ? |
| Pritumumab | | mab | human | vimentin | brain cancer |
| PRO 140 | | ? | humanized | CCR5 | HIV infection |
| Quilizumab[34] | | mab | humanized | IGHE | asthma |
| Tetulomab | | mab | humanized | CD37 | cancer[121] |
| Racotumomab[103] | | mab | mouse | N-glycolylneuraminic acid | cancer |
| Radretumab[20] | | mab | human | fibronectin extra domain-B | cancer |
| Rafivirumab[8] | | mab | human | rabies virus glycoprotein | rabies (prophylaxis) |
| Ralpancizumab[122] | | mab | humanized | neural apoptosis-regulated proteinase 1 | dyslipidemia |
| Ramucirumab | Cyramza | mab | human | VEGFR2 | solid tumors |
| Ranibizumab[6] | Lucentis | Fab | humanized | VEGF-A | macular degeneration (wet form) |
| Raxibacumab[23] | | mab | human | anthrax toxin, protective antigen | anthrax (prophylaxis and treatment) |
| Refanezumab[123] | | mab | humanized | myelin-associated glycoprotein | recovery of motor function after stroke |
| Regavirumab | | mab | human | cytomegalovirus glycoprotein B | cytomegalovirus infection |
| Reslizumab[52] | | mab | humanized | IL-5 | inflammations of the airways, skin and gastrointestinal tract |
| Rilotumumab[124] | | mab | human | HGF | solid tumors |
| Rinucumab[125] | | mab | human | platelet-derived growth factor receptor beta | neovascular age-related macular degeneration |
| Rituximab | MabThera, Rituxan | mab | chimeric | CD20 | lymphomas, leukemias, some autoimmune disorders |
| Robatumumab | | mab | human | IGF-1 receptor | cancer |
| Roledumab[76] | | mab | human | RHD | ? |
| Romosozumab[126] | | mab | humanized | sclerostin | osteoporosis |
| Rontalizumab[127] | | mab | humanized | IFN-α | systemic lupus erythematosus |
| Rovelizumab | LeukArrest | mab | humanized | CD11, CD18 | haemorrhagic shock etc. |
| Ruplizumab[11] | Antova | mab | humanized | CD154 (CD40L) | rheumatic diseases |
| Sacituzumab govitecan[128] | | mab | humanized | tumor-associated calcium signal transducer 2 | cancer |
| Samalizumab[129] | | mab | humanized | CD200 | cancer |
| Sarilumab[130] | | mab | human | IL6 | rheumatoid arthritis, ankylosing spondylitis |
| Satumomab pendetide | | mab | mouse | TAG-72 | cancer (diagnosis) |
| Secukinumab[131] | | mab | human | IL 17A | uveitis, rheumatoid arthritis psoriasis |
| Seribantumab[25] | | mab | human | ERBB3 | cancer |
| Setoxaximab[25] | | mab | chimeric | E. coli shiga toxin type-2 | ? |
| Sevirumab | | ? | human | cytomegalovirus | cytomegalovirus infection |
| Sibrotuzumab | | mab | humanized | FAP | cancer |
| SGN-CD19A | | mab | humanized | CD19 | acute lymphoblastic leukemia and B-cell non-Hodgkin lymphoma |
| SGN-CD33A | | mab | humanized | CD33 | Acute myeloid leukemia |
| Sifalimumab[132] | | mab | humanized | IFN-α | SLE, dermatomyositis, polymyositis |
| Siltuximab | | mab | chimeric | IL-6 | cancer |
| Simtuzumab[48] | | mab | humanized | LOXL2 | fibrosis |
| Siplizumab[16] | | mab | humanized | CD2 | psoriasis, graft-versus-host disease (prevention) |
| Sirukumab[133] | | mab | human | IL-6 | rheumatoid arthritis |
| Sofituzumab vedotin[134] | | mab | humanized | CA 125 | ovarian cancer |
| Solanezumab[103] | | mab | humanized | beta amyloid | Alzheimer's disease |
| Solitomab[34] | | mab | mouse | EpCAM | ? |
| Sonepcizumab[135] | | ? | humanized | sphingosine-1-phosphate | choroidal and retinal neovascularization |
| Sontuzumab[105] | | mab | humanized | episialin | ? |
| Stamulumab[42][105] | | mab | human | myostatin | muscular dystrophy |
| Sulesomab | LeukoScan | Fab' | mouse | NCA-90 (granulocyte antigen) | osteomyelitis (imaging) |
| Suvizumab[82] | | mab | humanized | HIV-1 | viral infections |
| Tabalumab[136] | | mab | human | BAFF | B-cell cancers |
| Tacatuzumab tetraxetan | AFP-Cide | mab | humanized | alpha-fetoprotein | cancer |
| Tadocizumab[105] | | Fab | humanized | integrin αIIbβ3 | percutaneous coronary intervention |
| Talizumab | | mab | humanized | IgE | allergic reaction |
| Tanezumab[8] | | mab | humanized | NGF | pain |
| Taplitumomab paptox[62] | | mab | mouse | CD19 | cancer |
| Tarextumab[137] | | mab | human | Notch receptor | cancer |
| Tefibazumab[23] | Aurexis | mab | humanized | clumping factor A | Staphylococcus aureus infection |
| Telimomab aritox | | Fab | mouse | ? | ? |
| Tenatumomab[9] | | mab | mouse | tenascin C | cancer |
| Teneliximab[16] | | mab | chimeric | CD40 | ? |
| Teplizumab[33] | | mab | humanized | CD3 | diabetes mellitus type 1 |
| Teprotumumab[138] | | mab | human | CD221 | hematologic tumors |
| Tesidolumab[19] | | mab | human | C5 | ? |
| TGN1412 | | ? | humanized | CD28 | chronic lymphocytic leukemia, rheumatoid arthritis |
| Ticilimumab (= tremelimumab) | | mab | human | CTLA-4 | cancer |
| Tildrakizumab[139] | | mab | humanized | IL23 | immunologically mediated inflammatory disorders |
| Tigatuzumab[9] | | mab | humanized | TRAIL-R2 | cancer |
| TNX-650 | | ? | humanized | IL-13 | Hodgkin's lymphoma |
| Tocilizumab[6] (= atlizumab) | Actemra, RoActemra | mab | humanized | IL-6 receptor | rheumatoid arthritis |
| Toralizumab[16] | | mab | humanized | CD154 (CD40L) | rheumatoid arthritis, lupus nephritis etc. |
| Tosatoxumab[3] | | mab | human | Staphylococcus aureus | ? |
| Tositumomab | Bexxar | ? | mouse | CD20 | follicular lymphoma |
| Tovetumab[140] | | mab | human | CD140a | cancer |
| Tralokinumab[141] | | mab | human | IL-13 | asthma etc. |
| Trastuzumab | Herceptin | mab | humanized | HER2/neu | breast cancer |
| Trastuzumab emtansine | Kadcyla | mab | humanized | HER2/neu | breast cancer |
| TRBS07[142] | Ektomab | 3funct | ? | GD2 | melanoma |
| Tregalizumab[20] | | mab | humanized | CD4 | ? |
| Tremelimumab | | mab | human | CTLA-4 | cancer |
| Trevogrumab[143] | | mab | human | growth differentiation factor 8 | muscle atrophy due to orthopedic disuse and sarcopenia |
| Tucotuzumab celmoleukin[42][105] | | mab | humanized | EpCAM | cancer |
| Tuvirumab | | ? | human | hepatitis B virus | chronic hepatitis B |
| Ublituximab[20] | | mab | chimeric | MS4A1 | cancer |
| Ulocuplumab[144] | | mab | human | C-X-C chemokine receptor type 4 | hematologic malignancies |
| Urelumab[145] | | mab | human | 4-1BB | cancer etc. |
| Urtoxazumab[6] | | mab | humanized | Escherichia coli | diarrhoea caused by E. coli |
| Ustekinumab[8] | Stelara | mab | human | IL-12, IL-23 | multiple sclerosis, psoriasis, psoriatic arthritis |
| Vandortuzumab vedotin[19] | | mab | humanized | STEAP1 | cancer |
| Vantictumab[146] | | mab | human | Frizzled receptor | cancer |
| Vanucizumab[22] | | mab | humanized | angiopoietin 2 | cancer |
| Vapaliximab[16] | | mab | chimeric | AOC3 (VAP-1) | ? |
| Varlilumab[147] | | mab | human | CD27 | ? |
| Vatelizumab[28] | | mab | humanized | ITGA2 | ? |
| Vedolizumab | | mab | humanized | integrin α4β7 | Crohn's disease, ulcerative colitis |
| Veltuzumab[9] | | mab | humanized | CD20 | non-Hodgkin's lymphoma |
| Vepalimomab | | mab | mouse | AOC3 (VAP-1) | inflammation |
| Vesencumab[20] | | mab | human | NRP1 | ? |
| Visilizumab[62] | Nuvion | mab | humanized | CD3 | Crohn's disease, ulcerative colitis |
| Volociximab[21] | | mab | chimeric | integrin α5β1 | solid tumors |
| Vorsetuzumab mafodotin[148] | | mab | humanized | CD70 | cancer |
| Votumumab | HumaSPECT | mab | human | tumor antigen CTAA16.88 | colorectal tumors |
| Zalutumumab[21] | HuMax-EGFr | mab | human | EGFR | squamous cell carcinoma of the head and neck |
| Zanolimumab[6] | HuMax-CD4 | mab | human | CD4 | rheumatoid arthritis, psoriasis, T-cell lymphoma |
| Zatuximab[48] | | mab | chimeric | HER1 | cancer |
| Ziralimumab[62] | | mab | human | CD147 (basigin) | ? |
| Zolimomab aritox | | mab | mouse | CD5 | systemic lupus erythematosus, graft-versus-host disease |