WIN 56,098

Systematic (IUPAC) name
anthracen-9-yl{2-methyl-1-[2-(morpholin-4-yl)ethyl]-1H-indol-3-yl}methanone
Identifiers
PubChem CID 9803721
ChemSpider 7979481
Chemical data
Formula C30H28N2O2
Molar mass 448.556 g/mol

WIN 56,098 is a chemical that is considered to be an aminoalkylindole derivative. It is a tricyclic aryl derivative that acts as a competitive antagonist at the CB2 cannabinoid receptor. Its activity at CB1 was significantly less effective. WIN 56,098 failed to antagonize any of the in vivo effects of THC.[1]

See also

References

  1. Howlett AC, Berglund B, Melvin LS (October 1995). "Cannabinoid Receptor Agonists and Antagonists". Current Pharmaceutical Design 1 (3): 343–352.


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