Etafedrine

Etafedrine
Systematic (IUPAC) name
(1R,2S)-2-[Ethyl(methyl)amino]-1-phenyl-1-propanol
Clinical data
Legal status
  • Withdrawn from market
Identifiers
CAS Number 7681-79-0 YesY
ATC code none
PubChem CID 10734
ChemSpider 85308 N
UNII 2Y6VQU63E8 YesY
Chemical data
Formula C12H19NO
Molar mass 193.285 g/mol
 NYesY (what is this?)  (verify)

Etafedrine (INN) or ethylephedrine is a long-acting bronchodilator and has the brand name Nethaprin. It was previously commercially available as both the free base and as the hydrochloride salt from Sanofi-Aventis (now Sanofi) but is now no longer marketed.

Pharmacology

Unlike ephedrine and tyramine, etafedrine does not induce the release of epinephrine or norepinephrine and instead acts as a selective β2 adrenoreceptor agonist, thereby mediating its bronchodilator effects.[1]

See also

References

  1. Lindmar, R; Löffelholz, K; Stieh-Koch, U (1985). "On the mechanism of bronchodilatation by etafedrine". Arzneimittel-Forschung 35 (3): 602–4. PMID 4039586.

This article is issued from Wikipedia - version of the Saturday, March 19, 2016. The text is available under the Creative Commons Attribution/Share Alike but additional terms may apply for the media files.