GAT100
 | |
| Systematic (IUPAC) name | |
|---|---|
|
3-ethyl-5-isothiocyanato-N-(4-(piperidin-1-yl)phenethyl)-1H-indole-2-carboxamide | |
| Chemical data | |
| Formula | C25H28N4OS |
| Molar mass | 432.58 g/mol |
GAT100 is a negative allosteric modulator of the cannabinoid CB1 receptor.[1][2]
See also
References
- ↑ "Novel Electrophilic and Photoaffinity Covalent Probes for Mapping the Cannabinoid 1 Receptor Allosteric Site(s).". doi:10.1021/acs.jmedchem.5b01303.
- ↑ "MAPPING CANNABINOID RECEPTOR 1 ALLOSTERIC SITE(S): CRITICAL MOLECULAR DETERMINANT AND SIGNALING PROFILE OF GAT100 - A NOVEL, POTENT AND IRREVERSIBLY BINDING PROBE.". doi:10.1021/acschemneuro.6b00041.
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