TC OT 39
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| Systematic (IUPAC) name | |
|---|---|
|
(2S)-N-[[4-[(4,10-dihydro-1-methylpyrazolo[3,4-b][1,5]benzodiazepin-5(1H)-yl)carbonyl]-2-methylphenyl]methyl]-2-[(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)thioxomethyl]-1-pyrrolidinecarboxamide | |
| Identifiers | |
| CAS Number | 479232-57-0 |
| ATC code | none |
| ChemSpider | 23249746 |
| Chemical data | |
| Formula | C32H40N8O2S |
| Molar mass | 600.78 g/mol |
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TC OT 39 is a non-peptide partial agonist of the oxytocin and vasopressin V2 receptors (Ki = 147 nM and >1000 nM, respectively) and antagonist of the vasopressin V1A receptor (Ki = 330 nM).[1]
See also
References
- ↑ Pitt GR, Batt AR, Haigh RM, Penson AM, Robson PA, Rooker DP, Tartar AL, Trim JE, Yea CM, Roe MB (September 2004). "Non-peptide oxytocin agonists". Bioorganic & Medicinal Chemistry Letters 14 (17): 4585–4589. doi:10.1016/j.bmcl.2004.04.107. PMID 15357997.
External links
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